Sercloremine
From Wikipedia, the free encyclopedia
![]() |
|
Names | |
---|---|
IUPAC name
4-(5-Chloro-1-benzofuran-2-yl)-1-methylpiperidine
|
|
Identifiers | |
54403-19-9 ![]() |
|
3D model (Jmol) | Interactive image |
ChemSpider | 142884 |
PubChem | 162749 |
|
|
|
|
Properties | |
C14H16ClNO | |
Molar mass | 249.74 g·mol−1 |
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
|
|
Infobox references | |
Sercloremine (CGP-4718A), usually as the hydrochloride salt, is a drug which was developed in the 1980s and was formerly under investigation as an antidepressant, but was never marketed.[1][2] It acts as a selective, reversible inhibitor of monoamine oxidase A (RIMA) and serotonin reuptake inhibitor.[1][3]
References[edit]
- ^ a b Barrie Hesp; Cain (2 September 1987). ANNUAL REPORTS IN MED CHEMISTRY V22 PPR. Academic Press. pp. 25–. ISBN 978-0-08-058366-2.
- ^ C.R. Ganellin; David J. Triggle (21 November 1996). Dictionary of Pharmacological Agents. CRC Press. pp. 1801–. ISBN 978-0-412-46630-4.
- ^ Delini-Stula, A.; Fischbach, R.; Gnirss, F.; Bures, E.; Pöldinger, W. (1985). "Early experience with CGP 4718 A (Sercloremine), a new selective and reversible MAO-A and 5-HT-uptake inhibitor, in the treatment of depressive patients". Drug Development Research. 6 (4): 371–384. doi:10.1002/ddr.430060409. ISSN 0272-4391.
![]() |
This drug article relating to the nervous system is a stub. You can help Wikipedia by expanding it. |