Cilobamine
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| Clinical data | |
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| ATC code | none |
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| CAS Number | 69429-84-1 |
| PubChem (CID) | 299379 |
| ChemSpider | 8557262 |
| UNII | 067U1T4S30  Y |
| ChEMBL | CHEMBL2106470 |
| Chemical and physical data | |
| Formula | C17H23Cl2NO |
| Molar mass | 328.27662 g/mol |
| 3D model (Jmol) | Interactive image |
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Cilobamine is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.[1][2]
It can clearly be seen that the structure is based on dichloroisoprenaline that has been fused onto the bicycloalkane scaffold.
See also[edit]
References[edit]
- ^ Leeson GA, Shaath ZA, Biedenbach SA, Yarrington JT, Okerholm RA. Dose related induction of the drug metabolizing enzymes of rat liver by cilobamine. Fundamental and Applied Toxicology. 1984 Apr;4(2 Pt 1):261-9. PMID 6724198
- ^ Wager, S.; Quitkin, F.; Stewart, J.; McGrath, P.; Harrison, W.; Markowitz, J.; Tricamo, E. (1988). "Cilobamine in the treatment of atypical depression". Human Psychopharmacology: Clinical and Experimental. 3 (3): 201. doi:10.1002/hup.470030308.
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