CP-1414S
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| Systematic (IUPAC) name | |
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1-phenyl-4-amino-8-nitro-3H-1,5-benzodiazepin-2-one
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| Identifiers | |
| CAS Number | 36975-99-2  |
| ATC code | none |
| PubChem | CID 37594 |
| ChemSpider | 34483 |
| Chemical data | |
| Formula | C15H12N4O3 |
| Molar mass | 296.280 g/mol |
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CP-1414S is an experimental drug first made by a team in Germany.[1] It is a benzodiazepine derivative. CP-1414S is a 1,5-benzodiazepine, with the nitrogen atoms located at positions 1 and 5 of the diazepine ring, and so is most closely related to other 1,5-benzodiazepines such as clobazam.
CP-1414S has primarily anxiolytic and anticonvulsant effects.[2] Its potency is roughly equal to that of clobazam, but with more pronounced sedation.[3]
See also[edit]
References[edit]
- ^ US 3766169
- ^ Carli M, Ballabio M, Caccia S, Garattini S, Samanin R (1981). "Studies on some pharmacological activities of 7-nitro-2-amino-5-phenyl-3H-1,5-benzodiazepine (CP 1414 S) in the rat. A comparison with diazepam". Arzneimittel-Forschung. 31 (10): 1721–3. PMID 6119091.
- ^ Mennini T, Garattini S (November 1982). "Benzodiazepine receptors': correlation with pharmacological responses in living animals". Life Sciences. 31 (19): 2025–35. doi:10.1016/0024-3205(82)90094-7. PMID 6129557.
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